Asymmetric synthesis of lysine analogues with reduced basicity, and their incorporation into proteasome inhibitors

Bruin, G. de; Rooden, E.J. van; Ward, D.; Wesseling, C.M.J.; Nieuwendijk, A.M.C.H. van den; Boeckel, C.A.A. van; ... ; Overkleeft, H.S. (2017)

Article / Letter to editor

• Asymmetric synthesis
• Amino acids
• Inhibitors
• Proteasomes
• Peptidomimetics
• Structure-activity relationships

• All authors: Bruin, G. de; Rooden, E.J. van; Ward, D.; Wesseling, C.M.J.; Nieuwendijk, A.M.C.H. van den; Boeckel, C.A.A. van; Driessen, C.; Kisselev, A.F.; Florea, B.I.; Stelt, M. van der; Overkleeft, H.S.
• Date: 2017-10-25
• Journal: European Journal of Organic Chemistry
• Volume: 2017
• Issue: 39
• Pages: 5921 - 5934
• DOI: doi:10.1002/ejoc.201701174