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Crystal structure and subsequent ligand design of a nonriboside partial agonist bound to the adenosine A2A receptor
Structural Mapping of Adenosine Receptor Mutations: Ligand Binding and Signaling Mechanisms
Kinetics for Drug Discovery: an industry-driven effort to target drug residence time
Controlling the dissociation of ligands from the adenosine A(2A) receptor through modulation of salt bridge strength