Proteasome inhibition and mechanism of resistance to a synthetic, library-based hexapeptide

Oerlemans, R.; Berkers, C.R.; Assaraf, Y.G.; Scheffer, G.L.; Peters, G.J.; Verbrugge, S.E.; ... ; Jansen, G. (2018)

Article / Letter to editor

• Proteasome
• Proteasome inhibitors
• Bortezomib
• Cytotoxic peptides
• Drug resistance
• ABC drug efflux transporters

• All authors: Oerlemans, R.; Berkers, C.R.; Assaraf, Y.G.; Scheffer, G.L.; Peters, G.J.; Verbrugge, S.E.; Cloos, J.; Slootstra, J.; Meloen, R.H.; Shoemaker, R.H.; Dijkmans, B.C.; Scheper, R.J.; Ovaa, H.; Jansen, G.
• Date: 2018-10-31
• Journal: Investigational New Drugs
• Volume: 36
• Issue: 5
• Pages: 797 - 809
• DOI: doi:10.1007/s10637-018-0569-x
• Link: https://link.springer.com/content/pdf/10.1007/s10637-018-0569-x.pdf