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Soethoudt, M.; Hoorens, M.W.H.; Doelman, W.; Martella, A.; Stelt, M. van der; Heitman, L.H. (2018)

Structure-kinetic relationship studies of cannabinoid CB2 receptor agonists reveal substituent-specific lipophilic effects on residence time

Article / Letter to editor
R agonists can be designed to have optimal kinetic profiles, which could aid the lead optimization process in drug discovery for the study or treatment of inflammatory diseases.
All authors
Soethoudt, M.; Hoorens, M.W.H.; Doelman, W.; Martella, A.; Stelt, M. van der; Heitman, L.H.
Date
2018-03-21
Journal
Biochemical pharmacology
Volume
152
Pages
129 - 142
DOI
doi:10.1016/j.bcp.2018.03.018