Incorporation of the Constrained Peptidomimetic, 5-Methylpyridin-2-one into Peptide Vinyl Sulfones and Peptide Epoxy Ketones is Detrimental for Proteasome Inhibition

Xin, B.T.; Bruin, G. de; Plomp, J.W.; Florea, B.I.; Marel, G.A. van der; Overkleeft, H.S. (2016)

Article / Letter to editor

• Medicinal chemistry
• Proteasome inhibitors
• Inhibitors
• Peptidomimetics
• Peptides

• All authors: Xin, B.T.; Bruin, G. de; Plomp, J.W.; Florea, B.I.; Marel, G.A. van der; Overkleeft, H.S.
• Date: 2016-02-28
• Issue: 6
• Pages: 1132 - 1144
• DOI: doi:10.1002/ejoc.201501401