Potent inhibition of nicotinamide N-methyltransferase by alkene linked bisubstrate mimics bearing electron deficient aromatics

Author(s):: Gao, Y.; Haren, M.J. van; Buijs, N.; Innocenti, P.; Zhang, Y.; Sartini, D.; Campagna, R.; Emanuelli, M.; Parsons, R.B.; Jespers, W.; Gutiérrez-de-Terán, H.; Westen, G.J.P. van (0000-0003-0717-1817); Martin, N.I.

Published: 2021
Publication type: Article / Letter to editor

Date issued: 2021-08-23
Language: English
Is part of: Journal of Medicinal Chemistry (2021), Vol. 64, no. 17, p. 12938–12963
hdl: 1887/3264236
doi: 10.1021/acs.jmedchem.1c01094