Incorporation of the Constrained Peptidomimetic, 5-Methylpyridin-2-one into Peptide Vinyl Sulfones and Peptide Epoxy Ketones is Detrimental for Proteasome Inhibition

Author(s):: Xin, B.T.; Bruin, G. de; Plomp, J.W.; Florea, B.I. (0000-0001-7114-2266); Marel, G.A. van der (0000-0001-8917-3458); Overkleeft, H.S. (0000-0001-6992-4760)

Published: 2016
Publication type: Article / Letter to editor

Medicinal chemistryProteasome inhibitorsInhibitorsPeptidomimeticsPeptides

Date issued: 2016-02-28
Language: English
Is part of
hdl: 1887/3199741
doi: 10.1002/ejoc.201501401