Asymmetric synthesis of lysine analogues with reduced basicity, and their incorporation into proteasome inhibitors

Author(s):
Bruin, G. de; Rooden, E.J. van (0000-0003-0041-6455); Ward, D.; Wesseling, C.M.J.; Nieuwendijk, A.M.C.H. van den; Boeckel, C.A.A. van; Driessen, C.; Kisselev, A.F.; Florea, B.I. (0000-0001-7114-2266); Stelt, M. van der (0000-0002-1029-5717); Overkleeft, H.S. (0000-0001-6992-4760)
Published
2017
Publication type
Article / Letter to editor
Asymmetric synthesisAmino acidsInhibitorsProteasomesPeptidomimeticsStructure-activity relationships
Date issued
2017-10-25
Language
English
Is part of
European Journal of Organic Chemistry (2017), Vol. 2017, no. 39, p. 5921-5934
hdl
1887/3192020
doi
10.1002/ejoc.201701174