The Alkyne Moiety as a Latent Electrophile in Irreversible Covalent Small Molecule Inhibitors of Cathepsin K

Author(s):
Mons, E.; Jansen, I.D.C.; Loboda, J.; Doodewaerd, B.R. van; Hermans, J.; Verdoes, M.; Boeckel, C.A.A. van; Veelen, P.A. van (0000-0002-7898-9408); Turk, B.; Turk, D.; Ovaa, H.
Published
2019
Publication type
Article / Letter to editor
Date issued
2019-02-27
Language
English
Is part of
Journal of the American Chemical Society (2019), Vol. 141, no. 8, p. 3507-3514
hdl
1887/120392
doi
10.1021/jacs.8b11027